Bisindolylmaleimide I HCl 176504-36-2
Bisindolylmaleimide I HCl
分子式:C25H24N4O2•HCl 分子量:448.94
产品描述
Bisindolylmaleimide I HCl是蛋白激酶C的抑制剂,也能够有效的抑制GSK-3
靶点
IC50
生物活性
An enhanced water-soluble form of Bisindolylmaleimide I.A reversible and ATP-competitive inhibitor of protein kinase C (Ki = 10 nM). May inhibit protein kinase A at much higher concentrations (Ki = 2 µM).
溶解性
DMSO 100 mM,水 10 mg/ml
稳定性
2年 -20°C粉状,6月-80°C溶于DMSO