Naloxone HCl dihydrate51481-60-8盐酸纳洛酮
盐酸纳洛酮
分子式:C19H21NO4.HCl.2(H2O) 分子量:399.87
产品描述
Naloxone HCl是阿片类反向激动剂药物,用于对抗阿片类药物过量的影响。
靶点
IC50
生物活性
Naloxone hydrochloride is a nonspecific opiate receptor antagonist that displays anitnociceptive effects. Studies have identified this product as a significant immunoadjuvant in cancer immunotherapy. Reportedly exhibits the ability to reverse various types of cardiovas Naloxone hydrochloride is an inhibitor of DOR, KOR, MOR and Sigma Receptor.
溶解性
DMSO 73 mg/mL,水 73 mg/mL,乙醇 <1 mg/mL
稳定性
2年 -20°C粉状,6月-80°C溶于DMSO